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Description: ETB antagonist
Biological Activity for IRL-1038
ETB endothelin receptor antagonist.
Technical Data for IRL-1038
| M. Wt | 1410 |
| Formula | C68H92N14O15S2 |
| Sequence |
CVYFCHLDIIW (Modifications: Disulfide bridge between 1 - 5) |
| Storage | Desiccate at -20°C |
| CAS Number | 144602-02-8 |
| PubChem ID | 16142511 |
| InChI Key | OETKRDJJNWJFOP-PJLZVMSOSA-N |
| Smiles | [H]N[C@H]1CSSC[C@H](NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@H](CC2=CC=C(O)C=C2)NC(=O)[C@@H](NC1=O)C(C)C)C(=O)N[C@@H](CC1=CNC=N1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CC1=CNC2=C1C=CC=C2)C(O)=O |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Product Datasheets for IRL-1038
References for IRL-1038
References are publications that support the biological activity of the product.
Haynes et al (1993) Endothelin; progress in pharmacology and physiology. TiPS 14 225 PMID: 8372400
Karaki et al (1993) ETB receptor antagonist, IRL 1038, selectively inhibits the endothelin-induced endothelium-dependent vascular relaxation. Eur.J.Pharmacol. 231 371 PMID: 8449230
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Keywords: IRL-1038, IRL-1038 supplier, ETB, antagonists, Receptors, Endothelin, 1195, Tocris Bioscience
1 Citation for IRL-1038
Citations are publications that use Tocris products. Selected citations for IRL-1038 include:
Khan et al (2006) Pharmacological characterization of endothelin receptors-mediated contraction in the mouse isolated proximal and distal colon. Br J Pharmacol 147 607 PMID: 16432510
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