BD 1008 dihydrobromide

Name: BD 1008 dihydrobromide
Brand: Tocris Bioscience
SKU: 0511

Cat. No. 0511 2 篇引用文献提交评论说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Discontinued Product

0511 has been discontinued.

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说明： Potent, selective σ ligand

化学名： N-[2-(3,4-Dichlorophenyl)ethyl]-N-methyl-2-(1-pyrrolidinyl)ethylamine dihydrobromide

说明书

引用文献 (2)

生物活性技术数据说明书参考文献

生物活性 for BD 1008 dihydrobromide

Potent and selective σ-ligand (K_i against [³H]-(+)-3-PPP = 0.34 nM).

技术数据 for BD 1008 dihydrobromide

分子量	463.08
公式	C₁₅H₂₂Cl₂N₂.2HBr
储存	Store at -20°C
CAS Number	138356-09-9
PubChem ID	45073417
InChI Key	YTBUMHOSKIAYCZ-UHFFFAOYSA-N
Smiles	Br.Br.CN(CCN1CCCC1)CCC1=CC=C(Cl)C(Cl)=C1

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

产品说明书 for BD 1008 dihydrobromide

分析证书/产品说明书

化学品安全技术说明书

参考文献 for BD 1008 dihydrobromide

参考文献是支持产品生物活性的出版物。

De Costa et al (1992) Synthesis, characterization, and biological evaluation of a novel class of N-(arylethyl)-N-alkyl-2-(1-pyrrolidinyl)ethylamines - structural requirements and binding affinity at the σ receptor. J.Med.Chem. 35 38 PMID: 1310114

Monnet et al (1996) Differentiation of σ ligand-activated receptor subtypes that modulate NMDA-evoked [³H]-noradrenaline release in rat hippocampal slices. Br.J.Pharmacol. 119 65 PMID: 8872358

Whittemore et al (1997) Antagonism of N-MthD.-aspartate receptors by σ site ligands: potency, subtype-selectivity and mechanisms of inhibition. J.Pharmacol.Exp.Ther. 282 326 PMID: 9223571

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关键词: BD 1008 dihydrobromide, BD 1008 dihydrobromide supplier, Potent, selective, σ, sigma, ligand, General, Receptors, BD1008, dihydrobromide, Sigma-Related, 0511, Tocris Bioscience

2 篇 BD 1008 dihydrobromide 的引用文献

引用文献是使用了 Tocris 产品的出版物。 BD 1008 dihydrobromide 的部分引用包括：

Hiranita et al (2011) Decreases in cocaine self-administration with dual inhibition of the DA transporter and σ receptors. J Pharmacol Exp Ther 339 662 PMID: 21859929

Hiranita et al (2013) Stimulants as specific inducers of DA-independentσ agonist self-administration in rats. Neurochem Int 347 42633 PMID: 23908387