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Submit ReviewBQ-3020
说明： Selective ETB agonist
纯度： ≥95% (HPLC)
生物活性 for BQ-3020
BQ-3020 is a highly potent and selective ETB endothelin receptor agonist (Ki values are 0.18 and 970 nM at human ETB and ETA receptors respectively).
技术数据 for BQ-3020
| 分子量 | 2006.35 |
| 公式 | C96H140N20O25S |
| 序列 |
LMDKEAVYFAHLDIIW (Modifications: Leu-1 = N-terminal Ac) |
| 储存 | Store at -20°C |
| 纯度 | ≥95% (HPLC) |
| CAS Number | 143113-45-5 |
| PubChem ID | 16135850 |
| InChI Key | AYJUXFCWNAVJLN-FHOIYVHLSA-N |
| Smiles | CC[C@H](C)[C@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC1=CNC=N1)NC(=O)[C@H](C)NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)[C@H](CC1=CC=C(O)C=C1)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCSC)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CC1=CNC2=C1C=CC=C2)C(O)=O |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
溶解性数据 for BQ-3020
| 溶解性 | Soluble to 0.50 mg/ml in sodium bicarbonate (0.03M) |
产品说明书 for BQ-3020
参考文献 for BQ-3020
参考文献是支持产品生物活性的出版物。
Ekelund et al (1994) Effects of selective ETB-receptor stimulation on arterial, venous and capillary functions in cat skeletal muscle. Br.J.Pharmacol. 112 887 PMID: 7921617
Ihara et al (1995) [3H]-BQ-123, a highly specific and reversible radioligand for the endothelin ETA receptor subtype. Eur.J.Pharmacol. 274 1 PMID: 7768260
Reynolds et al (1995) Pharmacological differences between rat and human endothelin B receptors. Biochem.Biophys.Res.Commun. 209 506 PMID: 7733918
Sakamoto et al (1993) Distinct subdomains of human endothelin receptors determine their selectivity to endothelinA-selective antagonist and endothelinB-selective agonists. J.Biol.Chem. 268 8547 PMID: 8473300
If you know of a relevant reference for BQ-3020, please let us know.
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关键词: BQ-3020, BQ-3020 supplier, Selective, ETB, agonists, Receptors, Endothelin, 1189, Tocris Bioscience
1 篇 BQ-3020 的引用文献
引用文献是使用了 Tocris 产品的出版物。 BQ-3020 的部分引用包括：
Hamby et al (2012) Inflammatory mediators alter the astrocyte transcriptome and calcium signaling elicited by multiple G-protein-coupled receptors. Cell Death Dis 32 14489 PMID: 23077035
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