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Submit ReviewCCG 63802
Discontinued Product
4028 has been discontinued.
View all Heterotrimeric G-protein GTPases products.
说明： Inhibitor of regulator of G-protein signaling 4 (RGS4) protein
化学名： (2E)-2-(1,3-Benzothiazol-2-yl)-3-[9-methyl-2-(3-methylphenoxy)-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl]acrylonitrile
纯度： ≥99% (HPLC)
生物活性 for CCG 63802
CCG 63802 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins. Selective amongst RGS proteins, with greatest potency at RGS4. Inhibits GTPase accelerating protein activity of RGS4 and blocks its interaction with Gαo. Retains activity under reducing conditions.
技术数据 for CCG 63802
| 分子量 | 450.51 |
| 公式 | C26H18N4O2S |
| 储存 | Store at +4°C |
| 纯度 | ≥99% (HPLC) |
| CAS Number | 620112-78-9 |
| PubChem ID | 6057678 |
| InChI Key | VFSVKVQMZDJFQX-NBVRZTHBSA-N |
| Smiles | O=C1C(/C=C(C#N)/C3=NC(C=CC=C4)=C4S3)=C(OC5=CC(C)=CC=C5)N=C2N1C=CC=C2C |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for CCG 63802
参考文献 for CCG 63802
参考文献是支持产品生物活性的出版物。
Blazer et al (2010) Reversible, allosteric small-molecule inhibitors of regulator of G protein signaling proteins. Mol.Pharmacol. 78 524 PMID: 20571077
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关键词: CCG 63802, CCG 63802 supplier, CCG63802, inhibitors, inhibits, regulator, g-protein, signaling, signalling, RGS, RGS4, G, proteins, Heterotrimeric, G-protein, GTPases, 4028, Tocris Bioscience
1 篇 CCG 63802 的引用文献
引用文献是使用了 Tocris 产品的出版物。 CCG 63802 的部分引用包括：
Taccola et al (2016) A new model of nerve injury in the rat reveals a role of Regulator of G protein Signaling 4 in tactile hypersensitivity. Experimental Neurology 286 1 PMID: 27641322
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