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Submit ReviewDeltorphin I
Discontinued Product
4591 has been discontinued.
说明： Potent δ agonist
生物活性 for Deltorphin I
Deltorphin I is a potent δ-opioid receptor agonist (IC50 = 0.5 nM in human granulocytes). Exhibits a high rate of blood-brain barrier penetrance.
技术数据 for Deltorphin I
| 分子量 | 768.87 |
| 公式 | C37H52N8O10 |
| 序列 |
YAFDVVG (Modifications: Ala-2 = D-Ala, Gly-7 = C-terminal amide) |
| 储存 | Store at -20°C |
| CAS Number | 122752-15-2 |
| PubChem ID | 10055958 |
| InChI Key | CJAORFIPPWIGPG-QXYJMILXSA-N |
| Smiles | [H]N[C@@H](CC1=CC=C(O)C=C1)C(=O)N[C@H](C)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C(C)C)C(=O)NCC(N)=O |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for Deltorphin I
参考文献 for Deltorphin I
参考文献是支持产品生物活性的出版物。
Stefano et al (1992) [D-Ala2]Deltorphin I binding and pharmacological evidence for a special subtype of δ opioid receptor on human and invertebrate immune cells. Proc.Natl.Acad.Sci.USA 89 9316 PMID: 1329092
Erspamer et al (1989) Deltorphins: a family of naturally occurring peptides with high affinity and selectivity for δ opioid binding sites. Proc.Natl.Acad.Sci.USA 86 5188 PMID: 2544892
Fiori et al (1997) Deltorphin transport across the blood-brain barrier. Proc.Natl.Acad.Sci.USA 94 9469 PMID: 9256506
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关键词: Deltorphin I, Deltorphin I supplier, DeltorphinI, delta, d, δ, opioids, agonists, brain, penetrant, bbb, Delta, Opioid, Receptors, 4591, Tocris Bioscience
1 篇 Deltorphin I 的引用文献
引用文献是使用了 Tocris 产品的出版物。 Deltorphin I 的部分引用包括：
Otis et al (2011) Spinal activation of delta opioid receptors alleviates cancer-related bone pain. Neuroscience 183 221 PMID: 21458544
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该领域的文献
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*请注意，Tocris 仅会向正规科研企业/机构地址发送文献。
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