Desmethyl-YM 298198

Discontinued Product

2447 has been discontinued.

View all Glutamate (Metabotropic) Group I Receptors products.
说明: Derivative of mGlu1 antagonist YM 298198 (Cat. No. 2448)
化学名: 6-Amino-N-cyclohexyl-3-methylthiazolo[3,2-a]benzimidazole-2-carboxamide hydrochloride
纯度: ≥98% (HPLC)
说明书
引用文献
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文献 (5)

生物活性 for Desmethyl-YM 298198

Desmethyl-YM 298198 is a derivative of the mGlu1-selective antagonist YM 298198 (Cat. No. 2448).

许可信息

Sold with the permission of Astellas Pharma Inc.

技术数据 for Desmethyl-YM 298198

分子量 364.89
公式 C17H20N4OS.HCl
储存 Desiccate at RT
纯度 ≥98% (HPLC)
CAS Number 1177767-57-5
PubChem ID 16759180
InChI Key SWKZWXJQIDXGLX-UHFFFAOYSA-N
Smiles Cl.CC1=C(SC2=NC3=CC=C(N)C=C3N12)C(=O)NC1CCCCC1

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

产品说明书 for Desmethyl-YM 298198

参考文献 for Desmethyl-YM 298198

参考文献是支持产品生物活性的出版物。

Kohara et al (2005) Radioligand binding properties and pharmacological characterization of 6-Amino-N-cyclohexyl-N,3-dimethyl-thiazolo[3,2-a]-benzimidazole-2-carboxamide (YM-298198), a high-affinity, selective and noncompetitive antagonist of metabo J.Pharmacol.Exp.Ther. 315 163 PMID: 15976016

关键词: Desmethyl-YM 298198, Desmethyl-YM 298198 supplier, Derivative, mGlu1, mGluR1, antagonists, YM, 298198, Group, I, Receptors, Glutamate, Metabotropic, Desmethyl-YM298198, (Metabotropic), 2447, Tocris Bioscience

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