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Estropipate

Cat. No. 3588 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Discontinued Product

3588 has been discontinued.

View all Estrogen and Related Receptors products.
说明： Estrogen receptor agonist and OATP1B1 inhibitor
化学名： Piperazine estrone sulfate
纯度： ≥97% (HPLC)
说明书
引用文献
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通路 (1)
生物活性 技术数据 说明书 参考文献

生物活性 for Estropipate

Estrogen receptor agonist. Also inhibits organic anion transporting polypeptide 1B1 (OATP1B1) (IC50= 70 nM).

技术数据 for Estropipate

分子量 436.56
公式 C18H22O5S.C4H10N2
储存 Store at RT
纯度 ≥97% (HPLC)
CAS Number 7280-37-7
PubChem ID 5284555
InChI Key HZEQBCVBILBTEP-ZFINNJDLSA-N
Smiles O=C4CC[C@@]3([H])[C@]2([H])CCC1=CC(OS(=O)(O)=O)=CC=C1[C@]([H])2CC[C@@]34C.C5NCCNC5

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

参考文献 for Estropipate

参考文献是支持产品生物活性的出版物。

Williams et al (2004) Estrogen regulation of the cytochrome P450 3A subfamily in humans. J.Pharmacol.Exp.Ther. 311 728 PMID: 15282264

Obaidat et al (2009) A cell-based high-throughput assay to identify inhibitors of organic anion transporting polypeptides 1B1 and 1B3. FASEB J. 23 748

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关键词: Estropipate, Estropipate supplier, Estrogen, receptor, agonists, OATP1B, inhibitors, inhibits, and, Related, Receptors, Multidrug, Transporters, 3588, Tocris Bioscience

⚠ WARNING: This product can expose you to chemicals including Estropipate, which is known to the State of California to cause reproductive toxicity with developmental effects. For more information, go to www.P65Warnings.ca.gov

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Pathways for Estropipate

Estrogen Signaling Pathway

Estrogen Signaling Pathway

Estrogen is a steroid hormone that is responsible for the regulation of growth, differentiation and function of the reproductive system. Estrogen signaling is often dysregulated in breast cancer and osteoporosis.