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Submit ReviewISAM 140
Discontinued Product
5965 has been discontinued.
View all Adenosine A<sub>2B</sub> Receptors products.
说明： High affinity A2B receptor antagonist
化学名： 4-(2-Furanyl)-4,10-dihydro-2-methylpyrimido[1,2-a]benzimidazole-3-carboxylic acid-1-methylethyl ester
纯度： ≥98% (HPLC)
生物活性 for ISAM 140
ISAM 140 is a high affinity A2B receptor antagonist (Ki = 3.49 nM). Exhibits >1000-fold selectivity for A2B over A1, A2A and A3 receptors.
技术数据 for ISAM 140
| 分子量 | 337.37 |
| 公式 | C19H19N3O3 |
| 储存 | Store at -20°C |
| 纯度 | ≥98% (HPLC) |
| CAS Number | 932191-62-3 |
| PubChem ID | 17198004 |
| InChI Key | NYHLRBMDXQBOIB-UHFFFAOYSA-N |
| Smiles | CC(OC(C1=C(N=C2NC3=CC=CC=C3N2C1C4=CC=CO4)C)=O)C |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for ISAM 140
参考文献 for ISAM 140
参考文献是支持产品生物活性的出版物。
El Maatougui et al (2016) Discovery of potent and highly selective A2B adenosine receptor antagonist chemotypes. J.Med.Chem. 59 1967 PMID: 26824742
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关键词: ISAM 140, ISAM 140 supplier, ISAM140, high, affinity, adenosine, receptors, A2B, selective, Adenosine, Receptors, 5965, Tocris Bioscience
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