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Submit ReviewMethimepip dihydrobromide
Discontinued Product
2947 has been discontinued.
View all Histamine H<sub>3</sub> Receptors products.
说明： Extremely selective H3 agonist
化学名： 4-(1H-Imidazol-4-ylmethyl)-1-methylpiperidine dihydrobromide
生物活性 for Methimepip dihydrobromide
Extremely selective histamine H3 receptor agonist (pKi values are 9.0, 5.7, < 5.0 and < 5.0 for hH3, hH4, hH1 and hH2 receptors respectively). Potently inhibits EFS-evoked contractions of guinea pig ileum (pD2 = 8.26).
技术数据 for Methimepip dihydrobromide
| 分子量 | 341.09 |
| 公式 | C10H17N3.2HBr |
| 储存 | Desiccate at RT |
| CAS Number | 817636-54-7 |
| PubChem ID | 11313836 |
| Smiles | CN1CCC(CC2=CNC=N2)CC1.Br.Br |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for Methimepip dihydrobromide
参考文献 for Methimepip dihydrobromide
参考文献是支持产品生物活性的出版物。
Kitbunnadaj et al (2005) N-substituted piperidinyl alkyl imidazoles: discovery of methimepip as a potent and selective histamine H3 receptor agonist. J.Med.Chem. 48 2100 PMID: 15771452
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关键词: Methimepip dihydrobromide, Methimepip dihydrobromide supplier, selective, H3, agonists, Receptors, Histamine, histaminergic, 2947, Tocris Bioscience
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该领域的文献
Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!
*请注意，Tocris 仅会向正规科研企业/机构地址发送文献。
Histamine Receptors Scientific Review
Written by Iwan de Esch and Rob Leurs, this review provides a synopsis of the different histamine receptor subtypes and the ligands that act upon them; compounds available from Tocris are listed.
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