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Submit ReviewNaltriben mesylate
Discontinued Product
0892 has been discontinued.
说明： Standard δ2 selective antagonist
化学名： 17-(Cyclopropylmethyl)-6,7-didehydro-3,14β-dihydroxy-4,5α-epoxy-6,7-2',3'-benzo[b]furanomorphinan mesylate
纯度： ≥98% (HPLC)
生物活性 for Naltriben mesylate
Naltriben mesylate is a selective and potent δ-opioid receptor antagonist (Ki values are 0.013, 19 and 152 nM for δ, μ and κ receptors respectively). Displays selectivity for the δ2 subtype in vivo.
许可信息
Sold with the permission of the University of Minnesota
技术数据 for Naltriben mesylate
| 分子量 | 511.59 |
| 公式 | C26H25NO4.CH3SO3H |
| 储存 | Desiccate at RT |
| 纯度 | ≥98% (HPLC) |
| CAS Number | 122517-78-6 |
| PubChem ID | 45073482 |
| InChI Key | XRRFZOCDAWPIBB-IDRHMUJXSA-N |
| Smiles | C[S](O)(=O)=O.[H][C@@]12OC3=C(O)C=CC4=C3[C@@]11CCN(CC3CC3)[C@]([H])(C4)[C@]1(O)CC1=C2OC2=C1C=CC=C2 |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for Naltriben mesylate
参考文献 for Naltriben mesylate
参考文献是支持产品生物活性的出版物。
Miyamoto et al (1993) Involvement of delta2 opioid receptors in the development of mor. dependence in mice. J.Pharmacol.Exp.Ther. 264 1141 PMID: 8383738
Portoghese et al (1991) Role of spacer and address components in peptidomimetic δ opioid receptor antagonists related to naltrindole. J.Med.Chem. 34 1715 PMID: 1851846
Thorat and Hammond (1997) Modulation of nociception by microinjection of delta-1 and delta-2 opioid receptor ligands in the ventromedial medulla of the rat. J.Pharmacol.Exp.Ther. 283 1185 PMID: 9399992
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关键词: Naltriben mesylate, Naltriben mesylate supplier, δ2-opioid, delta2-opioid, selective, antagonists, DOP, Receptors, OP1, Delta, Opioid, 0892, Tocris Bioscience
1 篇 Naltriben mesylate 的引用文献
引用文献是使用了 Tocris 产品的出版物。 Naltriben mesylate 的部分引用包括：
Gomes et al (2000) Heterodimerization of μ and δ opioid receptors: A role in opiate synergy. Exp Neurobiol 20 RC110 PMID: 11069979
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