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说明： Urotensin-II (UT) antagonist
生物活性 for UFP 803
UFP 803 is an urotensin-II (UT) receptor ligand; behaves as a silent antagonist in most in vitro assays and in vivo, but does retain small residual agonist activity under certain conditions in some assays. Competitively antagonizes U-II induced contractions in the rat aorta (pIC50 = 7.46) and prevents plasma extravasation elicited by U-II in mice in vivo.
技术数据 for UFP 803
| 分子量 | 1061.24 |
| 公式 | C50H64N10O12S2 |
| 序列 |
DXFWXYCV (Modifications: X-2 = Pen, Trp-4 = D-Trp, X-5 = Dab, Disulfide bridge between 2 - 7) |
| 储存 | Desiccate at -20°C |
| CAS Number | 879497-82-2 |
| PubChem ID | 90488769 |
| InChI Key | LRELVPJTCGYTSS-AAEZYUNISA-N |
| Smiles | [H]N[C@@H](CC(O)=O)C(=O)NC1C(=O)N[C@@H](CC2=CC=CC=C2)C(=O)N[C@H](CC2=CNC3=C2C=CC=C3)C(=O)NC(CCN)C(=O)N[C@@H](CC2=CC=C(O)C=C2)C(=O)N[C@@H](CSSC1(C)C)C(=O)N[C@@H](C(C)C)C(O)=O |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for UFP 803
参考文献 for UFP 803
参考文献是支持产品生物活性的出版物。
Camarda et al (2006) In vitro and in vivo pharmacological characterization of the novel UT receptor ligand [Pen5,DTrp7,Dab8]urotensin II(4-11) (UFP-803). Br.J.Pharmacol. 147 92 PMID: 16273120
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关键词: UFP 803, UFP 803 supplier, Urotensin, II, UT, antagonists, Receptors, Urotensin-II, UFP803, 2529, Tocris Bioscience
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