Zolantidine dimaleate

Cat. No. 1070 1 次引用提交评论说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

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说明： Potent, centrally active H₂ antagonist

化学名： N-[3-[3-(1-Piperidinylmethyl)phenoxy]propyl]-2-benzothiazolamine dimaleate

引用文献 (1)

文献 (1)

生物活性技术数据溶解性计算器说明书参考文献

生物活性 for Zolantidine dimaleate

Zolantidine dimaleate is a a potent, selective and brain penetrating H₂ receptor antagonist.

许可信息

Sold with the permission of GlaxoSmithKline

技术数据 for Zolantidine dimaleate

分子量	613.68
公式	C₂₂H₂₇N₃OS.2C₄H₄O₄
储存	Desiccate at +4°C
CAS Number	104076-39-3
PubChem ID	11957725
InChI Key	IECBEVAUEBZJCF-SPIKMXEPSA-N
Smiles	OC(=O)\C=C/C(O)=O.OC(=O)\C=C/C(O)=O.C(CNC1=NC2=C(S1)C=CC=C2)COC1=CC(CN2CCCCC2)=CC=C1

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

溶解性数据 for Zolantidine dimaleate

	溶剂	最高浓度 mg/mL	最高浓度 mM
溶解性
溶解性	water		100

制备储备液 for Zolantidine dimaleate

以下数据基于产品分子量 613.68。 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

浓度/溶剂体积/质量	1 mg	5 mg	10 mg
1 mM	1.63 mL	8.15 mL	16.3 mL
5 mM	0.33 mL	1.63 mL	3.26 mL
10 mM	0.16 mL	0.81 mL	1.63 mL
50 mM	0.03 mL	0.16 mL	0.33 mL

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产品说明书 for Zolantidine dimaleate

分析证书/产品说明书

化学品安全技术说明书

参考文献 for Zolantidine dimaleate

参考文献是支持产品生物活性的出版物。

Calcutt et al (1988) Zolantidine (SK&F 95282) is a potent selective brain penetrating histamine H₂-receptor antagonist. Br.J.Pharmacol. 93 69 PMID: 2894879

Coruzzi et al (1994) Activity of the new histamine H₂-receptor antagonist zolantidine at cardiac and gastric H₂ receptors. Pharmacology 48 69 PMID: 7907797

Coruzzi et al (1996) Cardiac and gastric effects of histamine H₂ receptor antagonists: no evidence for a correlation between lipophilicity and receptor affinity. Br.J.Pharmacol. 118 1813 PMID: 8842448

If you know of a relevant reference for Zolantidine dimaleate, please let us know.

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关键词: Zolantidine dimaleate, Zolantidine dimaleate supplier, Potent, centrally, active, H2, antagonists, Receptors, Histamine, histaminergic, GlaxoSmithKline, GSK, 1070, Tocris Bioscience

1 篇 Zolantidine dimaleate 的引用文献

引用文献是使用了 Tocris 产品的出版物。 Zolantidine dimaleate 的部分引用包括：

Porter et al (2005) Fenobam: a clinically validated nonbenzodiazepine anxiolytic is a potent, selective, and noncompetitive mGlu5 receptor antagonist with inverse agonist activity. J Pharmacol Exp Ther 315 711 PMID: 16040814

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