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Submit ReviewCarbetapentane citrate
Discontinued Product
0454 has been discontinued.
Description: High affinity σ1 ligand
Alternative Names: Pentoxyverine citrate
Chemical Name: 1-Phenylcyclopentanecarboxylic acid 2-(2-diethylaminoethoxy)ethyl ester citrate
Purity: ≥99% (HPLC)
Biological Activity for Carbetapentane citrate
Carbetapentane citrate is a selective ligand for the σ1 -site.
Technical Data for Carbetapentane citrate
| M. Wt | 525.59 |
| Formula | C20H31NO3.C6H8O7 |
| Storage | Store at RT |
| Purity | ≥99% (HPLC) |
| CAS Number | 23142-01-0 |
| PubChem ID | 90010 |
| InChI Key | AKJDEXBCRLOVTH-UHFFFAOYSA-N |
| Smiles | OC(=O)CC(O)(CC(O)=O)C(O)=O.CCN(CC)CCOCCOC(=O)C1(CCCC1)C1=CC=CC=C1 |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Product Datasheets for Carbetapentane citrate
References for Carbetapentane citrate
References are publications that support the biological activity of the product.
Quirion et al (1992) A proposal for the classification of sigma binding sites. TiPS 13 85 PMID: 1315463
Rothman et al (1991) Labelling by [3H]1,3-di(2-tolyl)guanidine of two high affinity binding sites in guinea pig brain: evidence for allosteric regulation by calcium channel antagonists and pseudoallosteric modulation by σ ligands. Mol.Pharmacol. 39 222 PMID: 1847495
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Keywords: Carbetapentane citrate, Carbetapentane citrate supplier, High, affinity, σ1, sigma1, ligand, Receptors, σ, sigma, selective, Pentoxyverine, citrate, Sigma1, 0454, Tocris Bioscience
1 Citation for Carbetapentane citrate
Citations are publications that use Tocris products. Selected citations for Carbetapentane citrate include:
Shin et al (2006) Vasoconstrictive neurovascular coupling during focal ischemic depolarizations. J Cereb Blood Flow Metab 26 1018 PMID: 16340958
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