(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

Name: (1 R ,1' S ,3' R /1 R ,1' R ,3' S )-L-054,264
Brand: Tocris Bioscience
SKU: 2444

Cat. No. 2444 提交评论说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Discontinued Product

2444 has been discontinued.

View all Somatostatin (sst) Receptors products.

说明： Potent and selective sst₂ agonist

化学名： N-[(1R)-2-[[[(1S*,3R*)-3-(Aminomethyl)cyclohexyl]methyl]amino]-1-(1H-indol-3-ylmethyl)-2-oxoethyl]spiro[1H-indene-1,4'-piperidine]-1'-carboxamide

纯度： ≥96% (HPLC)

说明书

引用文献

生物活性技术数据说明书参考文献

生物活性 for (1R,1'S,3'R/1R,1'R,3'S)-L-054,264

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 is a potent and selective somatostatin sst₂ receptor agonist (K_i values are 4, 537, 2480, 3614 and 5017 nM for cloned human sst₂, sst₁, sst₄, sst₃ and sst₅ receptors respectively).

技术数据 for (1R,1'S,3'R/1R,1'R,3'S)-L-054,264

分子量	539.71
公式	C₃₃H₄₁N₅O₂
储存	Store at +4°C
纯度	≥96% (HPLC)
CAS Number	208706-12-1
PubChem ID	9915239
InChI Key	DAMXHAMKVXERLM-FVBCXUTKSA-N
Smiles	NC[C@H]1CCC[C@@H](CNC([C@H](NC(N4CCC5(C(C=CC=C6)=C6C=C5)CC4)=O)CC2=CNC3=C2C=CC=C3)=O)C1

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

产品说明书 for (1R,1'S,3'R/1R,1'R,3'S)-L-054,264

分析证书/产品说明书

化学品安全技术说明书

参考文献 for (1R,1'S,3'R/1R,1'R,3'S)-L-054,264

参考文献是支持产品生物活性的出版物。

Yang et al (1998) Spiro[1H-indene-1,4'-piperidine] derivatives as potent and selective non-peptide human somatostatin receptor subtype 2 (sst₂) agonists. J.Med.Chem. 41 2175 PMID: 9632348

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关键词: (1R,1S,3R/1R,1R,3'S)-L-054,264, (1R,1S,3R/1R,1R,3'S)-L-054,264 supplier, Potent, selective, sst2, agonists, sst, Receptors, Somatostatin, (1R,1S,3R/1R,1R,3S)-L-054,264, L054264, 2444, Tocris Bioscience

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