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Submit ReviewBIM 23052
说明： sst5 agonist
生物活性 for BIM 23052
Somatostatin sst5 receptor agonist (Ki values are 7.3, 13.5, 31.3 and 141 nM for sst5, sst2, sst1 and sst4 receptors respectively). Stimulates gastric emptying following i.c. administration.
技术数据 for BIM 23052
| 分子量 | 1122.3 |
| 公式 | C61H75N11O10 |
| 序列 |
FFFWKTFT (Modifications: Phe-1 = D-Phe, Trp-4 = D-Trp, Thr-8 = C-terminal amide) |
| 储存 | Store at -20°C |
| CAS Number | 133073-82-2 |
| PubChem ID | 9963480 |
| InChI Key | HMTCBXPQKWFOMG-QWXJMLLVSA-N |
| Smiles | [H]N[C@H](CC1=CC=CC=C1)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@@H]([C@@H](C)O)C(N)=O |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for BIM 23052
参考文献 for BIM 23052
参考文献是支持产品生物活性的出版物。
Patel and Srikant (1994) Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstr 1-5). Endocrinology 135 2814 PMID: 7988476
Martinez et al (2000) Intracisternal injection of somatostatin receptor 5-preferring agonists induces a vagal cholinergic stimulation of gastric emptying in rats. J.Pharmacol.Exp.Ther. 293 1099 PMID: 10869415
Nunn et al (2002) Pharmacological characterisation of the goldfish somatostatin sst5 receptor. Eur.J.Pharmacol. 436 173 PMID: 11858797
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关键词: BIM 23052, BIM 23052 supplier, sst5, agonists, Receptors, Somatostatin, BIM23052, 2842, Tocris Bioscience
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