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BIM 23056

Cat. No. 1844 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Discontinued Product

1844 has been discontinued.

View all Somatostatin (sst) Receptors products.
说明： sst ligand
说明书
引用文献
评论
生物活性 技术数据 说明书 参考文献

生物活性 for BIM 23056

BIM 23056 is a somatostatin receptor ligand (Ki values are 142, > 1000, 10.8, 16.6 and 5.7 nM for human cloned sst1 - 5 receptors respectively). Behaves as an antagonist on SRIF14-induced [35S]-GTPγS binding at sst3 and sst5 receptors (PKB values are 6.33 and 5.84 respectively).

技术数据 for BIM 23056

分子量 1232.49
公式 C71H81N11O9
序列 FFYWKVFX

(Modifications: Phe-1 = D-Phe, Trp-4 = D-Trp, X = D-Nal & C-terminal amide)
储存 Desiccate at -20°C
CAS Number 150155-61-6
PubChem ID 16133799
InChI Key VPTPBEUWKCLZGU-OOSWLFMASA-N
Smiles [H]N[C@H](CC1=CC=CC=C1)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@@H](CC1=CC=C(O)C=C1)C(=O)N[C@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@H](CC1=CC2=CC=CC=C2C=C1)C(N)=O

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

产品说明书 for BIM 23056

分析证书/产品说明书
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化学品安全技术说明书目前不在网上提供。
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参考文献 for BIM 23056

参考文献是支持产品生物活性的出版物。

Patel and Srikant (1994) Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstr 1-5). Endocrinology 135 2814 PMID: 7988476

Raynor et al (1993) Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding of linear peptides. Mol.Pharmacol. 43 838 PMID: 8100350

Siehler and Hoyer (1999) Characterisation of human recombinant somatostatin receptors. Modulation of GTPgammaS binding. Naunyn Schmiedebergs Arch.Pharmacol. 360 500 PMID: 10598789

Wilkinson et al (1996) Potent antagonism by BIM-23056 at the human recombinant somatostatin sst5 receptor. Br.J.Pharmacol. 118 445 PMID: 8762063

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关键词: BIM 23056, BIM 23056 supplier, Somatostatin, receptor, agonists, Receptors, BIM23056, 1844, Tocris Bioscience

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