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CYM 50769

Cat. No. 4948 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）
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说明： Novel non-peptide NPBWR1 antagonist
别名： ML250
化学名： 5-Chloro-2-(9H-fluoren-9-yl)-4-(4-methoxyphenoxy)-3(2H)-pyridazinone
纯度： ≥98% (HPLC)
说明书
引用文献
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文献 (1)
生物活性 技术数据 溶解性 计算器 说明书 参考文献

生物活性 for CYM 50769

CYM 50769 is a novel non-peptide antagonist of neuropeptide W/B receptor 1 (NPBWR1, GPR7) (IC50 = 0.12 μM).

技术数据 for CYM 50769

分子量 416.86
公式 C24H17ClN2O3
储存 Store at +4°C
纯度 ≥98% (HPLC)
CAS Number 1421365-63-0
PubChem ID 50904505
InChI Key QHVSQUYCVUHYKT-UHFFFAOYSA-N
Smiles ClC(C=N4)=C(OC5=CC=C(OC)C=C5)C(N4C2C3=C(C=CC=C3)C1=CC=CC=C12)=O

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

溶解性数据 for CYM 50769

溶剂 最高浓度 mg/mL 最高浓度 mM
溶解性
DMSO 41.69 100

制备储备液 for CYM 50769

以下数据基于产品分子量 416.86。 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

选择批次从而根据批次分子量重新计算:
浓度/溶剂体积/质量 1 mg 5 mg 10 mg
1 mM 2.4 mL 11.99 mL 23.99 mL
5 mM 0.48 mL 2.4 mL 4.8 mL
10 mM 0.24 mL 1.2 mL 2.4 mL
50 mM 0.05 mL 0.24 mL 0.48 mL

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参考文献 for CYM 50769

参考文献是支持产品生物活性的出版物。

Guerrero et al (2013) SAR analysis of novel non-peptidic NPBWR1 (GPR7) antagonists. Bioorg.Med.Chem.Lett. 23 614 PMID: 23287738

If you know of a relevant reference for CYM 50769, please let us know.

按标靶查看相关产品

关键词: CYM 50769, CYM 50769 supplier, NPBWR1, antagonists, neuropeptide, B, W, receptor, 1, CYM50769, ML250, GPR7, Other, Peptide, Receptors, 4948, Tocris Bioscience

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