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Submit ReviewJNJ 1661010
说明： Selective, reversible FAAH inhibitor
化学名： N-Phenyl-4-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-piperazinecarboxamide
纯度： ≥99% (HPLC)
生物活性 for JNJ 1661010
JNJ 1661010 is a selective, reversible inhibitor of fatty acid amide hydrolase (FAAH) (IC50 = 12 nM). Brain penetrant and active in vivo.
技术数据 for JNJ 1661010
| 分子量 | 365.45 |
| 公式 | C19H19N5OS |
| 储存 | Store at +4°C |
| 纯度 | ≥99% (HPLC) |
| CAS Number | 681136-29-8 |
| PubChem ID | 2809273 |
| InChI Key | BHBOSTKQCZEAJM-UHFFFAOYSA-N |
| Smiles | O=C(NC3=CC=CC=C3)N1CCN(C2=NC(C4=CC=CC=C4)=NS2)CC1 |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for JNJ 1661010
参考文献 for JNJ 1661010
参考文献是支持产品生物活性的出版物。
Keith et al (2008) Thiadiazolopiperazinyl ureas as inhibitors of fatty acid amid hydrolase. Bioorg.Med.Chem.Lett. 18 4838 PMID: 18693015
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关键词: JNJ 1661010, JNJ 1661010 supplier, Selective, reversible, FAAH, inhibitors, inhibits, Anandamide, Amidase, Fatty, Acid, Amide, Hydrolases, JNJ1661010, Hydrolase, (FAAH), Other, Cannabinoids, 3262, Tocris Bioscience
2 篇 JNJ 1661010 的引用文献
引用文献是使用了 Tocris 产品的出版物。 JNJ 1661010 的部分引用包括：
Stone et al (2012) The cytoprotective effects of oleoylethanolamide in Ins-Secr.g cells do not require activation of GPR119. Br J Pharmacol 165 2758 PMID: 22029844
Brown et al (2010) Cannabinoid receptor-dependent and -independent anti-proliferative effects of omega-3 ethanolamides in androgen receptor-positive and -negative prostate cancer cell lines. Carcinogenesis 31 1584 PMID: 20660502
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