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Submit ReviewL-803,087 trifluoroacetate is a potent and selective somatostatin sst4 receptor agonist. Ki values are 0.7, 199, 4720, 1280 and 3880 nM for cloned human sst4, sst1, sst2, sst3 and sst5 receptors respectively. Facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice in vivo.
分子量 | 599.56 |
公式 | C25H29F2N5O3.CF3CO2H |
储存 | Store at -20°C |
纯度 | ≥97% (HPLC) |
CAS Number | 1786412-46-1 |
PubChem ID | 45073436 |
InChI Key | IIRYZHRNVKQVGQ-BDQAORGHSA-N |
Smiles | FC(F)(F)C(O)=O.NC(NCCC[C@@H]([C@@](OC)=O)NC(CCCC1=C(C3=CC=CC=C3)NC2=C1C=C(F)C=C2F)=O)=N |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
参考文献是支持产品生物活性的出版物。
Rohrer et al (1998) Rapid identification of subtype-selective agonists of the somatostatin receptor through combinatorial chemistry. Science 282 737 PMID: 9784130
Rohrer and Schaeffer (2000) Identification and characterization of subtype selective somatostatin receptor agonists. J.Physiol.Paris 94 211 PMID: 11087999
Moneta et al (2002) Somatostatin receptor subtypes 2 and 4 affect seizure susceptibility and hippocampal excitatory neurotransmission in mice. Eur.J.Neurosci. 16 843 PMID: 12372020
关键词: L-803,087 trifluoroacetate, L-803,087 trifluoroacetate supplier, Potent, selective, sst4, agonists, Receptors, Somatostatin, L803087, 1979, Tocris Bioscience
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