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[Orn5]-URP

Cat. No. 3162 1 次引用 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Discontinued Product

3162 has been discontinued.

View all Urotensin-II Receptors products.
说明： Urotensin-II (UT) receptor antagonist
说明书
引用文献 (1)
评论
生物活性 技术数据 说明书 参考文献

生物活性 for [Orn5]-URP

[Orn5]-URP is an urotensin-II (UT) receptor pure antagonist (pEC50 = 7.24). Displays no agonist activity unlike other U-II/URP analogs. Inhibits the action of U-II in the rat aorta ring assay.

技术数据 for [Orn5]-URP

分子量 1003.2
公式 C48H62N10O10S2
序列 ACFWXYCV

(Modifications: X = Orn, Disulfide bridge between 2 - 7)
储存 Store at -20°C
CAS Number 782485-03-4
PubChem ID 90488807
InChI Key BPLKRLYKWHXTMO-LSKWFVNGSA-N
Smiles [H]N[C@@H](C)C(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CC2=CC=C(O)C=C2)NC(=O)[C@H](CCCN)NC(=O)[C@H](CC2=CNC3=C2C=CC=C3)NC(=O)[C@H](CC2=CC=CC=C2)NC1=O)C(=O)N[C@@H](C(C)C)C(O)=O

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

参考文献 for [Orn5]-URP

参考文献是支持产品生物活性的出版物。

Chatenet et al (2004) Structure-activity relationships and structural conformation of a novel urotensin II-related peptide. Peptides 25 1819 PMID: 15476952

Diallo et al (2008) [Orn5]URP acts as a pure antagonist of urotensinergic receptors in rat cortical astrocytes. Peptides 29 813 PMID: 18082287

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关键词: [Orn5]-URP, [Orn5]-URP supplier, Urotensin-II, UT, receptor, antagonists, Receptors, 3162, Tocris Bioscience

1 篇 [Orn5]-URP 的引用文献

引用文献是使用了 Tocris 产品的出版物。 [Orn5]-URP 的部分引用包括：

Lee et al (2014) Urotensin II induces interleukin 8 expression in human umbilical vein endothelial cells. PLoS One 9 e90278 PMID: 24587311

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