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说明： sst2 and sst5 agonist
别名： MK 678
生物活性 for Seglitide
Peptide agonist for sst2 and sst5 somatostatin receptors. IC50/Kd values (nM) at cloned human somatostatin receptors are: > 1000 (sst1), 0.2 - 1.5 (sst2), 27 - 36 (sst3), > 127 (sst4), and 0.06 - 23 (sst5).
技术数据 for Seglitide
| 分子量 | 808.98 |
| 公式 | C44H56N8O7 |
| 序列 |
AYWKVF (Modifications: Ala-1 = N-methyl-Ala, Trp-3 = D-Trp, Cyclized) |
| 储存 | Desiccate at -20°C |
| CAS Number | 81377-02-8 |
| PubChem ID | 5311430 |
| InChI Key | NPJIOCBFOAHEDO-AVWFULIKSA-N |
| Smiles | CC(C)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CC2=CNC3=C2C=CC=C3)NC(=O)[C@H](CC2=CC=C(O)C=C2)NC(=O)[C@H](C)N(C)C(=O)[C@H](CC2=CC=CC=C2)NC1=O |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for Seglitide
参考文献 for Seglitide
参考文献是支持产品生物活性的出版物。
Hoyer et al (1994) Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch.Pharmacol. 350 441 PMID: 7870182
Raynor et al (1993) Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding to linear peptides. Mol.Pharmacol. 43 838 PMID: 8100350
Hannon et al (2002) Drug design at peptide receptors. Somatostatin receptor ligands. J.Mol.Neurosci. 18 15
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关键词: Seglitide, Seglitide supplier, sst2, sst5, agonists, Receptors, Somatostatin, MK678, MK, 678, 1836, Tocris Bioscience
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