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VUF 11207 fumarate

Cat. No. 4780 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Discontinued Product

4780 has been discontinued.

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说明： Potent ACKR3 (CXCR7) agonist
化学名： N-[(2E)-3-(2-Fluorophenyl)-2-methyl-2-propen-1-yl]-3,4,5-trimethoxy-N-[2-(1-methyl-2-pyrrolidinyl)ethyl]benzamide fumarate
纯度： ≥98% (HPLC)
说明书
引用文献
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文献 (1)
生物活性 技术数据 说明书 参考文献

生物活性 for VUF 11207 fumarate

VUF 11207 fumarate is a potent ACKR3 (CXCR7) chemokine receptor agonist (EC50 = 1.6 nM). Induces recruitment of β-arrestin to CXCR7 in HEK293-CXCR7 cells.

化合物库 for VUF 11207 fumarate

VUF 11207 fumarate is also offered as part of the Tocriscreen 2.0 Max. 了解 Tocris 化合物库的更多信息。

技术数据 for VUF 11207 fumarate

分子量 586.65
公式 C27H35FN2O4.C4H4O4
储存 Store at -20°C
纯度 ≥98% (HPLC)
CAS Number 1785665-61-3
PubChem ID 90488970
InChI Key MTPOECCHJLVVGO-FDULSSLPSA-N
Smiles C\C(CN(CCC2N(C)CCC2)C(C3=CC(OC)=C(OC)C(OC)=C3)=O)=C/C1=C(F)C=CC=C1.OC(/C=C/C(O)=O)=O

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

产品说明书 for VUF 11207 fumarate

分析证书/产品说明书
化学品安全技术说明书

参考文献 for VUF 11207 fumarate

参考文献是支持产品生物活性的出版物。

Wijtmans et al (2012) Synthesis, modeling and functional activity of substituted styrene-amides as small-molecule CXCR7 agonists. Eur.J.Med.Chem. 51 184 PMID: 22424612

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关键词: VUF 11207 fumarate, VUF 11207 fumarate supplier, VUF11207, fumarate, CXCR7, chemokine, receptors, potent, agonist, Chemokine, CXC, Receptors, 4780, Tocris Bioscience

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