GABAB Receptor Antagonists
| Cat. No. | Product Name / Activity |
|---|---|
| 1245 | CGP 35348 |
| Selective GABAB antagonist; brain penetrant | |
| 3219 | CGP 36216 hydrochloride |
| GABAB antagonist; displays activity at presynaptic receptors | |
| 1247 | CGP 46381 |
| Selective GABAB antagonist; brain penetrant | |
| 1246 | CGP 52432 |
| Potent and selective GABAB antagonist | |
| 1088 | CGP 54626 hydrochloride |
| Potent and selective GABAB antagonist | |
| 1248 | CGP 55845 hydrochloride |
| Potent and selective GABAB antagonist | |
| 0245 | 2-Hydroxysaclofen |
| Selective GABAB antagonist; more potent than Saclofen (Cat. No. 0246) | |
| 0246 | Saclofen |
| Selective GABAB antagonist | |
| 0984 | SCH 50911 |
| Selective and competitive GABAB antagonist; orally bioavailable |
GABA Scientific Review
Our GABA review gives an overview of the structure and function of the GABA receptors, as well as highlighting pharmacological ligands for their study.
Request copyRequest PDFAddiction Life Science Poster
Written by Prof David Nutt, this poster summarizes the brain circuits and neurotransmitter systems that are affected by the main classes of addictive drugs.
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