Submit a Review & Earn an Amazon Gift Card
You can now submit reviews for your favorite Tocris products. Your review will help other researchers decide on the best products for their research. Why not submit a review today?!
Submit ReviewBIM 23052
Description: sst5 agonist
Biological Activity for BIM 23052
Somatostatin sst5 receptor agonist (Ki values are 7.3, 13.5, 31.3 and 141 nM for sst5, sst2, sst1 and sst4 receptors respectively). Stimulates gastric emptying following i.c. administration.
Technical Data for BIM 23052
| M. Wt | 1122.3 |
| Formula | C61H75N11O10 |
| Sequence |
FFFWKTFT (Modifications: Phe-1 = D-Phe, Trp-4 = D-Trp, Thr-8 = C-terminal amide) |
| Storage | Store at -20°C |
| CAS Number | 133073-82-2 |
| PubChem ID | 9963480 |
| InChI Key | HMTCBXPQKWFOMG-QWXJMLLVSA-N |
| Smiles | [H]N[C@H](CC1=CC=CC=C1)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@@H]([C@@H](C)O)C(N)=O |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Product Datasheets for BIM 23052
References for BIM 23052
References are publications that support the biological activity of the product.
Patel and Srikant (1994) Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstr 1-5). Endocrinology 135 2814 PMID: 7988476
Martinez et al (2000) Intracisternal injection of somatostatin receptor 5-preferring agonists induces a vagal cholinergic stimulation of gastric emptying in rats. J.Pharmacol.Exp.Ther. 293 1099 PMID: 10869415
Nunn et al (2002) Pharmacological characterisation of the goldfish somatostatin sst5 receptor. Eur.J.Pharmacol. 436 173 PMID: 11858797
View Related Products by Target
View Related Products by Product Action
Keywords: BIM 23052, BIM 23052 supplier, sst5, agonists, Receptors, Somatostatin, BIM23052, 2842, Tocris Bioscience
Citations for BIM 23052
Citations are publications that use Tocris products.
Currently there are no citations for BIM 23052.
Reviews for BIM 23052
There are currently no reviews for this product. Be the first to review BIM 23052 and earn rewards!
Have you used BIM 23052?
Submit a review and receive an Amazon gift card.
$50/€35/£30/$50CAN/¥300 Yuan/¥5000 Yen for first to review with an image
$25/€18/£15/$25CAN/¥75 Yuan/¥2500 Yen for a review with an image
$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image