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Submit ReviewCilostazol
Description: PDE3A inhibitor. Also adenosine uptake inhibitor
Chemical Name: 6-[4-(1-Cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
Purity: ≥99% (HPLC)
Biological Activity for Cilostazol
Cilostazol is a potent phosphodiesterase III A (PDE3A) inhibitor (IC50 = 0.2 μM) and inhibitor of adenosine uptake. Has antimitogenic, antithrombotic, vasodilatory and cardiotonic properties in vivo. Also affects lipid levels in vivo.
Compound Libraries for Cilostazol
Cilostazol is also offered as part of the Tocriscreen 2.0 Max and Tocriscreen FDA-Approved Drugs. Find out more about compound libraries available from Tocris.
Technical Data for Cilostazol
| M. Wt | 369.47 |
| Formula | C20H27N5O2 |
| Storage | Store at RT |
| Purity | ≥99% (HPLC) |
| CAS Number | 73963-72-1 |
| PubChem ID | 2754 |
| InChI Key | RRGUKTPIGVIEKM-UHFFFAOYSA-N |
| Smiles | O=C1CCC2=CC(OCCCCC3=NN=NN3C3CCCCC3)=CC=C2N1 |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Product Datasheets for Cilostazol
References for Cilostazol
References are publications that support the biological activity of the product.
Schror (2002) The pharmacology of cilos. Diabetes Obes.Metab. 4 S14 PMID: 12180353
Shintani et al (1985) General pharmacological properties of cilostazol, a new antithrombotic drug. Part I: effects on the central nervous system. Arzneimittelforschung 35 1157 PMID: 4074429
Shintani et al (1985) General pharmacological properties of cilostazol, a new antithrombotic drug. Part II: effects on the peripheral organs. Arzneimittelforschung 35 1163 PMID: 3000392
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Keywords: Cilostazol, Cilostazol supplier, PDE3A, inhibitors, inhibits, adenosines, reuptake, Phosphodiesterases, ENT1, Purine, Transporters, Pyrimidine, Equilibrative, Nucleoside, Monoamine, Neurotransmitter, 1692, Tocris Bioscience
Citations for Cilostazol
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Currently there are no citations for Cilostazol.
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