Phosphodiesterase Inhibitors

Cat. No. Product Name / Activity
6313 A 33
Potent and selective PDE4B inhibitor
2237 BRL 50481
Selective PDE7 inhibitor
2793 Caffeine
Cyclic nucleotide PDE inhibitor
0915 Cilostamide
PDE3 inhibitor
0691 Dipyridamole
PDE5/6/8/10/11 inhibitor
1261 EHNA hydrochloride
PDE2 inhibitor
1693 Enoximone
PDE3 inhibitor
5202 Furamidine dihydrochloride
TDP-1 inhibitor; PRMT1 inhibitor
4165 Gisadenafil besylate
Potent PDE5 inhibitor; orally bioavailable
2845 IBMX
PDE inhibitor (non-selective)
1694 Ibudilast
PDE inhibitor (non-selective)
3053 Mesopram
Orally active PDE4 inhibitor
5915 PF 04449613
Potent PDE9 inhibitor; brain penetrant
6024 PF 04671536 hydrochloride
Potent and selective PDE8B/8A inhibitor
6405 PF 05180999
Potent and selective PDE2A inhibitor
4525 Piclamilast
Potent and selective PDE4 inhibitor
0415 Ro 20-1724
PDE4 inhibitor
0905 Rolipram
PDE4 inhibitor
1349 (R)-(-)-Rolipram
PDE4 inhibitor. More active enantiomer of rolipram (Cat. No. 0905)
3784 Sildenafil citrate
Potent PDE5 inhibitor; orally active
6311 Tadalafil
Potent and highly selective PDE5 inhibitor; orally bioavailable
2337 Trequinsin hydrochloride
Highly potent PDE3 inhibitor
0947 Zaprinast
PDE5/6/9/11 inhibitor