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Submit ReviewFentanyl citrate
Discontinued Product
3247 has been discontinued.
Description: Potent and selective μ agonist
Alternative Names: Phentanyl citrate
Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamide citrate
Purity: ≥99% (HPLC)
Biological Activity for Fentanyl citrate
Potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.
Technical Data for Fentanyl citrate
| M. Wt | 528.59 |
| Formula | C22H28N2O.C6H8O7 |
| Storage | Store at RT |
| Purity | ≥99% (HPLC) |
| CAS Number | 990-73-8 |
| PubChem ID | 13810 |
| InChI Key | IVLVTNPOHDFFCJ-UHFFFAOYSA-N |
| Smiles | O=C(O)C(O)(CC(O)=O)CC(O)=O.O=C(CC)N(C3=CC=CC=C3)C1CCN(CCC2=CC=CC=C2)CC1 |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Product Datasheets for Fentanyl citrate
References for Fentanyl citrate
References are publications that support the biological activity of the product.
Zernig et al (1995) Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding. Life Sci. 57 2113 PMID: 7475964
Liu et al (2003) Opioid activity of C8813, a novel and potent opioid analgesic. Life Sci. 73 233 PMID: 12738037
Stevenson et al (2003) Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception. J.Pharmacol.Exp.Ther. 307 1054 PMID: 14557380
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Currently there are no citations for Fentanyl citrate.
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