Meptazinol hydrochloride

Discontinued Product

3636 has been discontinued.

Description: μ1 partial agonist
Chemical Name: 3-(3-Ethylhexahydro-1-methyl-1H-azepin-3-yl)phenol hydrochloride
Purity: ≥99% (HPLC)
Datasheet
Citations
Reviews
Literature (2)

Biological Activity for Meptazinol hydrochloride

Meptazinol hydrochloride is a centrally active opioid analgesic. Partial agonist at the μ1 opioid receptor. Also shown to inhibit acetylcholinesterase.

Technical Data for Meptazinol hydrochloride

M. Wt 269.81
Formula C15H23NO.HCl
Storage Desiccate at +4°C
Purity ≥99% (HPLC)
CAS Number 59263-76-2
PubChem ID 65483
InChI Key MPJUSISYVXABBH-UHFFFAOYSA-N
Smiles OC1=CC=CC(C2(CC)CN(C)CCCC2)=C1.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for Meptazinol hydrochloride

Certificate of Analysis / Product Datasheet
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References for Meptazinol hydrochloride

References are publications that support the biological activity of the product.

Spiegel and Pasternak (1984) Meptazinol: a novel Mu-1 selective opioid analgesic. J.Pharmacol.Exp.Ther. 228 414 PMID: 6141283

Galli et al (1996) Reversible inhibition of cholinesterases by opioids: possible pharmacological consequences. J.Pharm.Pharmacol. 48 116

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Keywords: Meptazinol hydrochloride, Meptazinol hydrochloride supplier, Partial, agonists, μ1-opioid, mu1-opioid, Receptors, MOP, OP3, μ-opioid, mu-opioid, Mu, Opioid, 3636, Tocris Bioscience

Citations for Meptazinol hydrochloride

Citations are publications that use Tocris products.

Currently there are no citations for Meptazinol hydrochloride.

Reviews for Meptazinol hydrochloride

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Literature in this Area

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!

*Please note that Tocris will only send literature to established scientific business / institute addresses.


Peptides Involved in Appetite Modulation Scientific Review

Peptides Involved in Appetite Modulation Scientific Review

Written by Sonia Tucci, Lynsay Kobelis and Tim Kirkham, this review provides a synopsis of the increasing number of peptides that have been implicated in appetite regulation and energy homeostasis; putative roles of the major peptides are outlined and compounds available from Tocris are listed.

Addiction Poster

Addiction Poster

The key feature of drug addiction is the inability to stop using a drug despite clear evidence of harm. This poster describes the brain circuits associated with addiction, and provides an overview of the main classes of addictive drugs and the neurotransmitter systems that they target.