8-Cyclopentyl-1,3-dimethylxanthine

Cat. No. 6137 提交评论说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Pricing	Availability		Qty

说明： High affinity adenosine A₁ receptor antagonist

别名： CPT,8-Cyclopentyltheophylline

化学名： 8-Cyclopentyltheophylline

纯度： ≥99% (HPLC)

生物活性技术数据溶解性计算器说明书参考文献

生物活性 for 8-Cyclopentyl-1,3-dimethylxanthine

8-Cyclopentyl-1,3-dimethylxanthine is a high affinity adenosine A₁ receptor antagonist (pKi = 7.5-8).

化合物库 for 8-Cyclopentyl-1,3-dimethylxanthine

8-Cyclopentyl-1,3-dimethylxanthine is also offered as part of the Tocriscreen 2.0 Max. 了解 Tocris 化合物库的更多信息。

技术数据 for 8-Cyclopentyl-1,3-dimethylxanthine

分子量	248.28
公式	C₁₂H₁₆N₄O₂
储存	Store at RT
纯度	≥99% (HPLC)
CAS Number	35873-49-5
PubChem ID	1917
InChI Key	SCVHFRLUNIOSGI-UHFFFAOYSA-N
Smiles	CN1C2=C(C(N(C1=O)C)=O)N=C(C3CCCC3)N2

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

溶解性数据 for 8-Cyclopentyl-1,3-dimethylxanthine

	溶剂	最高浓度 mg/mL	最高浓度 mM
溶解性
	DMSO	24.83	100
	ethanol	2.48	10

制备储备液 for 8-Cyclopentyl-1,3-dimethylxanthine

以下数据基于产品分子量 248.28。 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

浓度/溶剂体积/质量	1 mg	5 mg	10 mg
1 mM	4.03 mL	20.14 mL	40.28 mL
5 mM	0.81 mL	4.03 mL	8.06 mL
10 mM	0.4 mL	2.01 mL	4.03 mL
50 mM	0.08 mL	0.4 mL	0.81 mL

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产品说明书 for 8-Cyclopentyl-1,3-dimethylxanthine

分析证书/产品说明书

化学品安全技术说明书

参考文献 for 8-Cyclopentyl-1,3-dimethylxanthine

参考文献是支持产品生物活性的出版物。

Dalpiaz et al (1998) Thermodynamics of full agonist, partial agonist, and antagonist binding to wild-type and mutant adenosine A₁ receptors. Biochem.Pharmacol. 56 1437 PMID: 9827575

If you know of a relevant reference for 8-Cyclopentyl-1,3-dimethylxanthine, please let us know.

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关键词: 8-Cyclopentyl-1,3-dimethylxanthine, 8-Cyclopentyl-1,3-dimethylxanthine supplier, Adenosine, A1, receptors, antagonists, antagonism, high, affinity, CPT, 8-Cyclopentyltheophylline, Receptors, 6137, Tocris Bioscience

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