主页 / 药理学 / Enzymes / Proteases / Aminopeptidases / Aminopeptidase Inhibitors / Bestatin

Bestatin

Cat. No. 1956 1 条评论 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）
Pricing Availability   Qty
说明： Aminopeptidase inhibitor
别名： Ubenimex
化学名： N-[(2S,3R)-3-Amino-2-hydroxy-1-oxo-4-phenylbutyl]-L-leucine
纯度： ≥98% (HPLC)
说明书
引用文献
评论 (1)
生物活性 技术数据 溶解性 计算器 说明书 参考文献

生物活性 for Bestatin

Bestatin is an aminopeptidase inhibitor (Ki = 0.001 - 90 mM); inhibits enkephalin metabolism and leukotriene A4 hydrolase. Inhibits tumor cell proliferation.

技术数据 for Bestatin

分子量 308.38
公式 C16H24N2O4
储存 Store at +4°C
纯度 ≥98% (HPLC)
CAS Number 58970-76-6
PubChem ID 72172
InChI Key VGGGPCQERPFHOB-RDBSUJKOSA-N
Smiles CC(C)C[C@H](NC(=O)[C@@H](O)[C@H](N)CC1=CC=CC=C1)C(O)=O

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

溶解性数据 for Bestatin

溶剂 最高浓度 mg/mL 最高浓度 mM
溶解性
1eq. NaOH 3.08 10

制备储备液 for Bestatin

以下数据基于产品分子量 308.38。 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

选择批次从而根据批次分子量重新计算:
浓度/溶剂体积/质量 1 mg 5 mg 10 mg
0.1 mM 32.43 mL 162.14 mL 324.28 mL
0.5 mM 6.49 mL 32.43 mL 64.86 mL
1 mM 3.24 mL 16.21 mL 32.43 mL
5 mM 0.65 mL 3.24 mL 6.49 mL

Molarity Calculator

Calculate the mass, volume, or concentration required for a solution.
=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and CoA (available online).

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Dilution Calculator

Calculate the dilution required to prepare a stock solution.
x
=
x

产品说明书 for Bestatin

分析证书/产品说明书
选择另一批次：
化学品安全技术说明书

参考文献 for Bestatin

参考文献是支持产品生物活性的出版物。

Imamura and Kimura (2000) Effect of ubenimex (Bestatin) on the cell growth and phenotype of HL-60 and HL-60R cell lines: up- and down-regulation of CD13/aminopeptidase N. Leuk.Lymphoma 37 663 PMID: 11042531

Scornik and Botbol (2001) Bestatin as an experimental tool in mammals. Curr.Drug Metab. 2 67 PMID: 11465152

Umezawa et al (1976) Bestatin, an inhibitor of aminopeptidase B, produced by actinomycetes. J.Antibiot. 29 97 PMID: 931798

If you know of a relevant reference for Bestatin, please let us know.

按标靶查看相关产品

按产品操作查看相关产品

查看全部 Aminopeptidase Inhibitors

关键词: Bestatin, Bestatin supplier, Aminopeptidase, inhibitors, inhibits, enkephalin, metabolism, leukotrienes, eicosanoids, A4, hydrolase, Proteases, Proteinases, Ubenimex, Aminopeptidases, LTA4, Hydrolase, 1956, Tocris Bioscience

篇 Bestatin 的引用文献

引用文献是使用了 Tocris 产品的出版物。

目前没有 Bestatin 的引用文献。 您是否知道使用了 Tocris Bestatin 的优秀论文？ 请告知我们.

Bestatin 的评论

平均评分: 5 (Based on 1 Review.)

5 星
100%
4 星
0%
3 星
0%
2 星
0%
1 星
0%

Have you used Bestatin?

Submit a review and receive an Amazon gift card.

$50/€35/£30/$50CAN/¥300 Yuan/¥5000 Yen for first to review with an image

$25/€18/£15/$25CAN/¥75 Yuan/¥2500 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review

Filter by:


Works well. Recommended..
By Anonymous on 05/14/2019
分析类型： Ex Vivo
种属： Mouse

Used for slice electrophysiology work; bath applied with the opioid peptide dynorphin A to prevent its degradation with great results.

review image