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Cilostazol

Cat. No. 1692 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）
Pricing Availability   Qty
说明： PDE3A inhibitor. Also adenosine uptake inhibitor
化学名： 6-[4-(1-Cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
纯度： ≥99% (HPLC)
说明书
引用文献
评论
生物活性 技术数据 溶解性 计算器 说明书 参考文献

生物活性 for Cilostazol

Cilostazol is a potent phosphodiesterase III A (PDE3A) inhibitor (IC50 = 0.2 μM) and inhibitor of adenosine uptake. Has antimitogenic, antithrombotic, vasodilatory and cardiotonic properties in vivo. Also affects lipid levels in vivo.

化合物库 for Cilostazol

Cilostazol is also offered as part of the Tocriscreen 2.0 Max and Tocriscreen FDA-Approved Drugs. 了解 Tocris 化合物库的更多信息。

技术数据 for Cilostazol

分子量 369.47
公式 C20H27N5O2
储存 Store at RT
纯度 ≥99% (HPLC)
CAS Number 73963-72-1
PubChem ID 2754
InChI Key RRGUKTPIGVIEKM-UHFFFAOYSA-N
Smiles O=C1CCC2=CC(OCCCCC3=NN=NN3C3CCCCC3)=CC=C2N1

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

溶解性数据 for Cilostazol

溶剂 最高浓度 mg/mL 最高浓度 mM
溶解性
ethanol 3.69 10
DMSO 18.47 50

制备储备液 for Cilostazol

以下数据基于产品分子量 369.47。 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

选择批次从而根据批次分子量重新计算:
浓度/溶剂体积/质量 1 mg 5 mg 10 mg
0.5 mM 5.41 mL 27.07 mL 54.13 mL
2.5 mM 1.08 mL 5.41 mL 10.83 mL
5 mM 0.54 mL 2.71 mL 5.41 mL
25 mM 0.11 mL 0.54 mL 1.08 mL

Molarity Calculator

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Reconstitution Calculator

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Dilution Calculator

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参考文献 for Cilostazol

参考文献是支持产品生物活性的出版物。

Schror (2002) The pharmacology of cilos. Diabetes Obes.Metab. 4 S14 PMID: 12180353

Shintani et al (1985) General pharmacological properties of cilostazol, a new antithrombotic drug. Part I: effects on the central nervous system. Arzneimittelforschung 35 1157 PMID: 4074429

Shintani et al (1985) General pharmacological properties of cilostazol, a new antithrombotic drug. Part II: effects on the peripheral organs. Arzneimittelforschung 35 1163 PMID: 3000392

If you know of a relevant reference for Cilostazol, please let us know.

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关键词: Cilostazol, Cilostazol supplier, PDE3A, inhibitors, inhibits, adenosines, reuptake, Phosphodiesterases, ENT1, Purine, Transporters, Pyrimidine, Equilibrative, Nucleoside, Monoamine, Neurotransmitter, 1692, Tocris Bioscience

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