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JWH 133 (in Tocrisolve™ 100)

Cat. No. 1783 1 次引用 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Discontinued Product

1783 has been discontinued.

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说明： Potent, selective CB2 agonist (in water-soluble emulsion)
化学名： (6aR,10aR)-3-(1,1-dimethylbutyl)-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran
说明书
引用文献 (1)
评论
文献 (1)
生物活性 技术数据 说明书 参考文献

生物活性 for JWH 133 (in Tocrisolve™ 100)

Potent CB2 selective agonist (Ki = 3.4 nM), in water-soluble emulsion (for details see TocrisolveTM 100). Approx. 200-fold selective over CB1 receptors. Active in vivo, reducing spasticity in a murine model of multiple sclerosis.

JWH 133 available as a solid.

技术数据 for JWH 133 (in Tocrisolve™ 100)

分子量 312.49
公式 C22H32O
储存 Store at +4°C
CAS Number 259869-55-1
PubChem ID 6918505
InChI Key YSBFLLZNALVODA-RBUKOAKNSA-N
Smiles [H][C@]([C@]3([H])C(C)(C)O2)(CC(C)=CC3)C1=C2C=C(C(C)(C)CCC)C=C1

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

产品说明书 for JWH 133 (in Tocrisolve™ 100)

分析证书/产品说明书
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化学品安全技术说明书

参考文献 for JWH 133 (in Tocrisolve™ 100)

参考文献是支持产品生物活性的出版物。

Baker et al (2000) Cannabinoids control spasticity and tremor in a multiple sclerosis model. Nature 404 84 PMID: 10716447

Huffman et al (1999) 3-(1'-Dimethylbutyl)-1-deoxy-Δ8-THC and related compounds: synthesis of selective ligands for the CB2 receptor. Bioorg.Med.Chem. 7 2905 PMID: 10658595

Pertwee (1999) Pharmacology of cannabinoid receptor ligands. Curr.Med.Chem. 6 635 PMID: 10469884

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关键词: JWH 133 (in Tocrisolve 100), JWH 133 (in Tocrisolve 100) supplier, Potent, selective, CB2, agonists, water-soluble, emulsion, cannabinoids, Receptors, JWH133, cb2r, 1783, Tocris Bioscience

1 篇 JWH 133 (in Tocrisolve™ 100) 的引用文献

引用文献是使用了 Tocris 产品的出版物。 JWH 133 (in Tocrisolve™ 100) 的部分引用包括：

Williams et al (2014) △(9)-Tetrahydrocannabinol treatment during human monocyte differentiation reduces macrophage susceptibility to HIV-1 infection. Autophagy 9 369 PMID: 24562630

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该领域的文献

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!

*请注意，Tocris 仅会向正规科研企业/机构地址发送文献。

Cannabinoid Receptor Ligands Scientific Review

Cannabinoid Receptor Ligands Scientific Review

Written by Roger Pertwee, this review discusses compounds which affect the activity of the endocannabinoid system, focusing particularly on ligands that are most widely used as experimental tools and denotes compounds available from Tocris.