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SLIGKV-NH2

Cat. No. 3010 1 次引用 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）
Pricing Availability   Qty
说明： PAR2 receptor agonist
纯度： ≥95% (HPLC)
说明书
引用文献 (1)
评论
生物活性 技术数据 溶解性 计算器 说明书 参考文献

生物活性 for SLIGKV-NH2

SLIGKV-NH2 is a protease-activated receptor 2 (PAR2) agonist (Ki = 9.64 μM and IC50 = 10.4 μM). Corresponds to the tethered ligand exposed by trypsin cleavage of PAR-2.

Control Peptide also available.

技术数据 for SLIGKV-NH2

分子量 614.78
公式 C28H54N8O7
序列 SLIGKV

(Modifications: Val-6 = C-terminal amide)
储存 Store at -20°C
纯度 ≥95% (HPLC)
CAS Number 190383-13-2
PubChem ID 10483914
InChI Key HOWDUIVVWDUEED-WAUHAFJUSA-N
Smiles [H]N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C(C)C)C(N)=O

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

溶解性数据 for SLIGKV-NH2

溶解性 Soluble to 1 mg/ml in water

产品说明书 for SLIGKV-NH2

分析证书/产品说明书
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化学品安全技术说明书

参考文献 for SLIGKV-NH2

参考文献是支持产品生物活性的出版物。

Bohm et al (1996) Molecular cloning, expression and potential functions of the human proteinase-activated receptor-2. Biochem.J. 314 1009 PMID: 8615752

Hollenberg and Compton (2002) International union of pharmacology XXVIII. Proteinase-activated receptors. Pharmacol.Rev. 54 203 PMID: 12037136

Kanke et al (2005) Binding of a highly potent protease-activated receptor-2 (PAR2) activating peptide, [3H]2-furoyl-LIGRL-NH2, to human PAR2. Br.J.Pharmacol. 145 255 PMID: 15765104

If you know of a relevant reference for SLIGKV-NH2, please let us know.

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关键词: SLIGKV-NH2, SLIGKV-NH2 supplier, PAR2, receptor, agonists, Receptors, Protease-Activated, proteinase-activated, 3010, Tocris Bioscience

1 篇 SLIGKV-NH2 的引用文献

引用文献是使用了 Tocris 产品的出版物。 SLIGKV-NH2 的部分引用包括：

Namkung et al (2016) Monitoring G protein-coupled receptor and [beta]-arrestin trafficking in live cells using enhanced bystander BRET Nature Communications 7 12178 PMID: 27397672

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