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TC-G 1001

Cat. No. 4879 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）
Pricing Availability   Qty
说明： GPR35 agonist; more potent than zaprinast (Cat. No. 0947)
化学名： 4-[[2-[(2-Fluorophenyl)amino]-4-oxo-5(4H)-thiazolylidene]methyl]benzoic acid
纯度： ≥98% (HPLC)
说明书
引用文献
评论
生物活性 技术数据 溶解性 计算器 说明书 参考文献

生物活性 for TC-G 1001

TC-G 1001 is a GPR35 agonist (pEC50 values are 7.59 and 8.36 for β-arrestin and Gαq-i5 Ca2+ assays respectively). Displays 1000-fold greater potency at human GPR35 receptors relative to mouse and rat GPR35 orthologs in an IP1 accumulation assay. More potent than zaprinast (Cat. No. 0947).

技术数据 for TC-G 1001

分子量 342.34
公式 C17H11FN2O3S
储存 Store at +4°C
纯度 ≥98% (HPLC)
CAS Number 494191-73-0
PubChem ID 5766343
InChI Key SYCKPHBALHXMIR-ZROIWOOFSA-N
Smiles O=C1N=C(NC3=CC=CC=C3F)S/C1=C\C2=CC=C(C(O)=O)C=C2

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

溶解性数据 for TC-G 1001

溶剂 最高浓度 mg/mL 最高浓度 mM
溶解性
DMSO 3.42 10

制备储备液 for TC-G 1001

以下数据基于产品分子量 342.34。 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

选择批次从而根据批次分子量重新计算:
浓度/溶剂体积/质量 1 mg 5 mg 10 mg
0.1 mM 29.21 mL 146.05 mL 292.11 mL
0.5 mM 5.84 mL 29.21 mL 58.42 mL
1 mM 2.92 mL 14.61 mL 29.21 mL
5 mM 0.58 mL 2.92 mL 5.84 mL

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参考文献 for TC-G 1001

参考文献是支持产品生物活性的出版物。

Neetoo-Isseljee et al (2013) High-throughput identification and characterization of novel, species-selective GPR35 agonists. J.Pharmacol.Exp.Ther. 344 568 PMID: 23262279

If you know of a relevant reference for TC-G 1001, please let us know.

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关键词: TC-G 1001, TC-G 1001 supplier, TC-G1001, GPR35, G, protein, coupled, receptor, 35, agonists, selective, 4879, Tocris Bioscience

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