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Submit ReviewTegaserod maleate
说明： 5-HT4 partial agonist
化学名： 2-[(5-Methoxy-1H-indol-3-yl)methylene]-N-pentyl-hydrazinecarboximidamide maleate
纯度： ≥99% (HPLC)
生物活性 for Tegaserod maleate
Tegaserod maleate is a partial agonist of 5-HT4 (Ki = 12 nM).
技术数据 for Tegaserod maleate
| 分子量 | 417.46 |
| 公式 | C16H23N5O.C4H4O4 |
| 储存 | Store at +4°C |
| 纯度 | ≥99% (HPLC) |
| CAS Number | 189188-57-6 |
| PubChem ID | 135413539 |
| InChI Key | CPDDZSSEAVLMRY-FEQFWAPWSA-N |
| Smiles | O=C(/C=C\C(O)=O)O.CCCCCNC(N/N=C/C1=CNC2=C1C=C(OC)C=C2)=N |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for Tegaserod maleate
参考文献 for Tegaserod maleate
参考文献是支持产品生物活性的出版物。
Buchheit et al (1995) The serotonin 5-HT4 receptor. 2. Structure-activity studies of the indole carbazimidamide class of agonists. J.Med.Chem. 38 2331 PMID: 7608899
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关键词: Tegaserod maleate, Tegaserod maleate supplier, Tegaserod, maleate, partial, 5-HT4, agonists, serotonergics, Receptors, 4613, Tocris Bioscience
1 篇 Tegaserod maleate 的引用文献
引用文献是使用了 Tocris 产品的出版物。 Tegaserod maleate 的部分引用包括：
Beattie et al (2011) The Pharmacology of TD-8954, a Potent and Selective 5-HT(4) Receptor Agonist with Gastrointestinal Prokinetic Properties. Front Pharmacol 2 25 PMID: 21687517
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该领域的文献
Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!
*请注意，Tocris 仅会向正规科研企业/机构地址发送文献。
5-HT Receptors Scientific Review
Written by Nicholas M. Barnes and John F. Neumaier, this review summarizes the various serotonin receptor subtypes and their importance in mediating the role of serotonin in numerous physiological and pharmacological processes. Compounds available from Tocris are listed.
Depression Poster
Major depressive disorder is characterized by depressed mood and a loss of interest and/or pleasure. Updated in 2015 this poster highlights presynaptic and postsynaptic targets for the potential treatment of major depressive disorder, as well as outlining the pharmacology of currently approved antidepressant drugs.