Cat. No. |
Product Name / Activity |
6712 |
A 77-01 |
| Potent inhibitor of TGF-βRI |
2939 |
A 83-01 |
| Selective inhibitor of TGF-βRI, ALK4 and ALK7 |
6870 |
AZ 12799734 |
| Potent TGF-βRI inhibitor |
2902 |
D 4476 |
| TGF-βRI inhibitor. Also inhibits CK1 |
6956 |
Galunisertib |
| ALK4 and ALK5 (TGFβRI) inhibitor |
3264 |
GW 788388 |
| Potent and selective inhibitor of TGF-βRI |
6016 |
IN 1130 |
| Potent and selective inhibitor of TGF-βRI |
7864 |
LY 2109761 |
| Selective TGF-β kinase inhibitor |
5288 |
R 268712 |
| Potent and selective inhibitor of TGF-βRI |
3742 |
RepSox |
| Potent and selective inhibitor of TGF-βRI |
1614 |
SB 431542 |
| Potent, selective inhibitor of TGF-βRI, ALK4 and ALK7 |
3263 |
SB 505124 |
| Selective inhibitor of TGF-βRI, ALK4 and ALK7 |
3211 |
SB 525334 |
| Selective inhibitor of TGF-βRI |
3269 |
SD 208 |
| Potent ATP-competitive TGF-βRI inhibitor |
6245 |
SM 16 |
| Potent TGF-βRI inhibitor; orally bioavailable |