| Cat. No. |
Product Name / Activity |
| 5781 |
A 425619 |
| Potent TRPV1 antagonist |
| 4319 |
A 784168 |
| Potent and selective TRPV1 antagonist |
| 4330 |
AMG 21629 |
| Potent and selective TRPV1 antagonist |
| 5995 |
AMG 517 |
| Potent TRPV1 antagonist |
| 2316 |
AMG 9810 |
| Potent and selective TRPV1 competitive antagonist |
| 3875 |
BCTC |
| TRPV1 antagonist |
| 0464 |
Capsazepine |
| TRPV antagonist; also activator of ENaCδ |
| 7199 |
(±)-Eriodictyol |
| Potent TRPV1 antagonist; also antioxidant; activates Nrf2/ARE signaling |
| 5106 |
GSK 2193874 |
| Potent and selective TRPV4 antagonist; orally active |
| 4100 |
HC 067047 |
| Potent and selective TRPV4 antagonist |
| 3361 |
JNJ 17203212 |
| Reversible, competitive and potent TRPV1 antagonist |
| 3746 |
RN 1734 |
| Selective TRPV4 antagonist |
| 5678 |
RN 9893 hydrochloride |
| Potent and selective TRPV4 antagonist |
| 1439 |
Ruthenium Red |
| Blocks capsaicin-activated cation channels |
| 1615 |
SB 366791 |
| Potent and selective TRPV1 competitive antagonist |
| 6990 |
SET 2 |
| Selective TRPV2 antagonist |
| 1098 |
Tranilast |
| Antiallergic; inhibits TRPV2-mediated responses |
| 6831 |
TRPV3 74a |
| Selective TRPV3 antagonist; brain penetrant |