Filter Results
Products (393)
Targets (4)
Resources (4)

"pharmacology" has 393 results in Products.

Results per Page:

PSEM 308 hydrochloride

Cat. No. 6425/5
Description: PSAML141F-GlyR and PSAML141F,Y115F-5-HT3 chimeric ion channel agonist
Purity: ≥98% (HPLC)
Pricing & Availability Qty

PSEM 89S

Cat. No. 6426/5
Description: PSAML141F-GlyR and PSAML141F,Y115F-5-HT3 chimeric ion channel agonist
Purity: ≥98% (HPLC)
Pricing & Availability Qty

Pexacerfont

Cat. No. 6451/10
Description: Potent and selective CRF1 antagonist; anxiolytic
Purity: ≥98% (HPLC)
Pricing & Availability Qty

PF 06551600 malonate

Cat. No. 6506/5
Description: Potent and selective JAK3 inhibitor
Purity: ≥98% (HPLC)
Pricing & Availability Qty

MLN 4924

Cat. No. 6499/10
Description: Potent and selective NEDD8 activating enzyme (NAE) inhibitor; cell permeable
Purity: ≥98% (HPLC)
Pricing & Availability Qty

AACOCF3

Cat. No. 1462/5
Description: Phospholipase A2 inhibitor
Pricing & Availability Qty

Vemurafenib

Cat. No. 7309/10
Description: Potent BRAF and CRAF inhibitor
Purity: ≥98% (HPLC)
Pricing & Availability Qty

Adavosertib

Cat. No. 7589/10
Description: Potent and selective Wee1 inhibitor
Purity: ≥98% (HPLC)
Pricing & Availability Qty

8-Bromo-cAMP, sodium salt

Cat. No. 1140/10
Description: Cell-permeable cAMP analog
Purity: ≥99% (HPLC)
Pricing & Availability Qty

R 7050

Cat. No. 5432/10
Description: Inhibitor of TNF-α receptor 1 signaling
Purity: ≥98% (HPLC)
Pricing & Availability Qty
Pageof 40

"pharmacology" has 4 results in Targets.

Chemogenetics

Chemogenetics is a powerful and specific method to control and investigate intracellular signaling pathways. Most widely used in neuroscience to control neuronal or glial cell activity, chemogenetic experiments employ compounds that selectively target a genetically-modified G protein-coupled receptor (GPCR; DREADD) or a chimeric ion channel (PSAM).

More Info

PSEMs

Pharmacologically Selective Effector Molecules (PSEMs) are inert ligands, specific for genetically-modified, chimeric ion channels, termed Pharmacologically Selective Actuator Modules (PSAMs). PSAMs containing the 5-HT3 ion pore domain allow activation of neuronal activity, while GlyR and GABAc containing chimeras are inhibitory

More Info

Pharmacology

Pharmacology is the study of interactions between drugs and biological systems. It is also the study of drug sources and their intrinsic properties. Most drugs act on defined pharmacological targets in order to exert their effects. The term drug is intended to mean any substance that alters normal biochemical function. Drugs with medicinal properties are termed pharmaceuticals.

Tocris products are categorised according to pharmacological activity. Click on any link below for further information.

More Info

"pharmacology" has 4 results in Resources.

Allosteric GPCR Pharmacology Poster

G protein-coupled receptors (GPCRs) are intrinsically allosteric proteins. This poster provides insights into allosteric mechanisms of GPCR biology, highlighting key facets of GPCR allostery and therapeutic applications of allosteric modulators.

More Info

Browse the Tocris Product Range by Pharmacological Activity

View and buy high purity products active at a range of pharmacological targets from Tocris Bioscience, the leading worldwide supplier of high performance life science reagents.

More Info

Chemogenetics Research Bulletin

Produced by Tocris, the chemogenetics research bulletin provides an introduction to chemogenetic methods to manipulate neuronal activity. It outlines the development of RASSLs, DREADDs and PSAMs, and the use of chemogenetic compounds. DREADD ligands and PSEMs available from Tocris are highlighted.

More Info

GPCR Efficacy and Biased Agonism Life Science Poster

GPCRs can interact with multiple distinct transducers or regulatory proteins and these can be preferentially engaged in an agonist-specific manner giving rise to biased agonism. This poster discusses cutting edge GPCR signaling pharmacology and highlights therapeutic applications of biased agonism.

More Info
Back to Search Results
Apply
Filters Clear All
Categories
Show More