Histamine H1 Receptor Antagonists

Cat. No. 产品名称/活性
3489 Astemizole
Orally active, potent H1 antagonist; also KV11.1 (hERG) channel blocker
1453 Clemastine fumarate
H1 antagonist
1425 (S)-(+)-Dimethindene maleate
H1 antagonist. Also M2 muscarinic antagonist
3072 Diphenhydramine hydrochloride
H1 antagonist
4245 Meclizine dihydrochloride
H1 antagonist; human pregnane X receptor agonist
2018 Mirtazapine
Potent H1 antagonist; also 5-HT2, 5-HT3 and α2 antagonist; antidepressant
4241 Olopatadine hydrochloride
H1 antagonist; ocular antiallergic agent
3948 Terfenadine
H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker