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CID 2011756

Cat. No. 4644 Submit a Review Datasheet / COA / SDS

Discontinued Product

4644 has been discontinued.

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Description: Pan protein kinase D (PKD) inhibitor; cell permeable
Chemical Name: 5-(3-Chlorophenyl)-N-[4-(4-morpholinylmethyl)phenyl]-2-furancarboxamide
Purity: ≥99% (HPLC)
Datasheet
Citations
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Biological Activity Technical Data Datasheets References

Biological Activity for CID 2011756

CID 2011756 is a protein kinase D (PKD) inhibitor (IC50 values are 0.6, 0.7 and 3.2 μM for PKD2, PKD3 and PKD1 respectively). Cell permeable (EC50 = 10 μM for PKD1 inhibition). ATP-competitive.

Technical Data for CID 2011756

M. Wt 396.87
Formula C22H21ClN2O3
Storage Store at RT
Purity ≥99% (HPLC)
CAS Number 638156-11-3
PubChem ID 2011756
InChI Key XQJWTJLJEYIUDZ-UHFFFAOYSA-N
Smiles O=C(NC3=CC=C(CN4CCOCC4)C=C3)C1=CC=C(C2=CC=CC(Cl)=C2)O1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

References for CID 2011756

References are publications that support the biological activity of the product.

Sharlow et al (2011) Discovery of diverse small molecule chemotypes with cell-based PKD1 inhibitory activity. PLoS One 6 e25134 PMID: 21998636

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Citations for CID 2011756

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Currently there are no citations for CID 2011756.

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