κ Opioid Receptor Agonists

Cat. No. Product Name / Activity
0699 BRL 52537 hydrochloride
Potent and selective κ agonist
3195 Dynorphin A
Endogenous κ agonist
1483 GR 89696 fumarate
Subtype-selective κ agonist
7541 Helianorphin-19
Potent and selective G protein-biased κ opioid receptor (KOR) agonist
0778 ICI 199,441 hydrochloride
Potent κ agonist
0822 ICI 204,448 hydrochloride
κ agonist, acts peripherally
0471 (+)-U-50488 hydrochloride
Selective κ agonist; less active enantiomer of (±)-U-50488 (Cat. No. 0495)
0495 (±)-U-50488 hydrochloride
Selective κ agonist
0496 (-)-U-50488 hydrochloride
Selective κ agonist; more active enantiomer of (±)-U-50488 (Cat. No. 0495)