|
Cat. No. |
产品名称/活性 |
5141 |
AZD 5582 dihydrochloride |
| Dimeric Smac mimetic; potent IAP inhibitor |
6955 |
Ceapin A7 |
| Selective inhibitor of ATF6α; sensitizes cells to ER stress |
3922 |
Eeyarestatin I |
| Potent inhibitor of ER-associated protein degradation and translocation |
5284 |
trans-ISRIB |
| Integrated stress response (ISR) inhibitor |
5153 |
ML 240 |
| ATP-competitive inhibitor of p97 ATPase |
6180 |
NMS 873 |
| Potent and selective p97 ATPase (VCP) allosteric inhibitor |
2347 |
Salubrinal |
| Selective inhibitor of eIF2a dephosphorylation |
4825 |
TC ASK 10 |
| Potent and selective ASK1 inhibitor; orally bioavailable |
4686 |
Xanthohumol |
| p97 ATPase (VCP) inhibitor |
|
Cat. No. |
产品名称/活性 |
4515 |
2-Deoxy-D-glucose |
| Enhances chimeric antigen receptor T cell activity. Disrupts N-glycan expression |
|
Cat. No. |
产品名称/活性 |
1231 |
Brefeldin A |
| Disrupts Golgi apparatus resulting in activation of ER stress pathways |
5869 |
CDN 1163 |
| SERCA2 allosteric activator |
7192 |
SMIP 004 |
| S-phase kinase-associated protein 2 (SKP2) inhibitor; activates UPR |
Other |
Cat. No. |
产品名称/活性 |
6759 |
AA 147 |
| ER proteostasis regulator |
1072 |
AGN 192403 hydrochloride |
| Binds TMED9 cargo receptor; releases mutant MUC-1 from vesicles and promotes trafficking to lysosome fro degradation |
6116 |
BHPI |
| Activates unfolded protein response; also ERα antagonist |