NMDA Receptor Antagonists

Cat. No.	产品名称/活性
3693	DL-AP5 Sodium salt
	Potent and selective NMDA antagonist; sodium salt of DL-AP5
0106	D-AP5
	Potent and selective NMDA receptor antagonist; more active form of DL-AP5
0105	DL-AP5
	Potent and selective NMDA antagonist
0107	L-AP5
	Potent and selective NMDA antagonist; less active form of DL-AP5
4492	Cerestat
	Potent and noncompetitive NMDA antagonist
1469	CGP 37849
	Potent and selective NMDA antagonist
1493	CGP 78608 hydrochloride
	Potent and selective NMDA antagonist; acts at glycine site
1241	CGS 19755
	Potent competitive NMDA antagonist
3697	7-Chlorokynurenic acid sodium salt
	Sodium salt of 7-Chlorokynurenic acid
0237	7-Chlorokynurenic acid
	NMDA antagonist; acts at glycine site
0190	CNQX
	NMDA antagonist; acts at glycine site; also AMPA/kainate antagonist
2456	Co 101244 hydrochloride
	GluN2B-selective NMDA antagonist
0247	(R)-CPP
	Potent NMDA antagonist; more active enantiomer of (RS)-CPP
0173	(RS)-CPP
	Potent NMDA antagonist
1265	D-CPP-ene
	Potent competitive NMDA antagonist
0286	5,7-Dichlorokynurenic acid
	Potent NMDA antagonist; acts at glycine site
3698	5,7-Dichlorokynurenic acid sodium salt
	Potent NMDA antagonist, acts at glycine site; sodium salt of 5,7-Dichlorokynurenic acid
4491	DQP 1105
	GluN2C/GluN2D-selective NMDA antagonist
2867	Flupirtine maleate
	Indirect NMDA antagonist; also GABA_A modulator and K_v7 channel activator
2348	Gavestinel
	Potent and selective NMDA antagonist; acts at the glycine site
0545	Ifenprodil hemitartrate
	Non-competitive NMDA antagonist; also σ ligand
3131	Ketamine hydrochloride
	Non-competitive NMDA antagonist
6751	(R)-(-)-Ketamine hydrochloride
	NMDA antagonist; antidepressant; may not display psychotomimetic or addictive side effects of (S)-ketamine
4379	(S)-(+)-Ketamine hydrochloride
	NMDA antagonist; enantiomer of ketamine hydrochloride
0742	L-689,560
	Highly potent NMDA antagonist
0705	L-701,252
	NMDA antagonist; acts at glycine site
0907	L-701,324
	NMDA antagonist; acts at glycine site
0840	Loperamide hydrochloride
	NMDA antagonist; reduces Ca²⁺ flux
0773	Memantine hydrochloride
	NMDA antagonist; acts at ion channel site
0924	(+)-MK 801 maleate
	Non-competitive NMDA antagonist; acts at ion channel site
0955	(-)-MK 801 maleate
	NMDA antagonist; less active enantiomer of (+)-MK 801
1970	Norketamine hydrochloride
	Potent non-competitive NMDA antagonist; antinociceptive
5018	PEAQX tetrasodium salt
	Potent and GluN2A-selective NMDA antagonist
2557	Phencyclidine hydrochloride
	Non-competitive NMDA antagonist
2530	PPDA
	GluN2C/GluN2D-selective NMDA antagonist
4801	QNZ 46
	Non-competitive and GluN2C/GluN2D-selective NMDA antagonist
1594	Ro 25-6981 maleate
	GluN2B-selective NMDA antagonist
3254	Ro 61-8048
	NMDA antagonist; increases kynurenic acid levels
4154	TCN 201
	GluN1/GluN2A-selective NMDA antagonist