All Products

Displaying Products by Catalog Number (4800 - 4899)

Cat. No. Product Name / Activity
4800 4EGI-1
Inhibits eIF4E:eIF4G subunit interaction
4801 QNZ 46
Non-competitive and GluN2C/GluN2D-selective NMDA antagonist
4803 CRANAD 2
Near-infrared probe that detects Aβ40 aggregates. Used for: amyloid-β detection in vitro and in vivo. Application: fluorescence microscopy, epifluorescence microscopy
4804 APETx2
ASIC3 channel blocker
4806 BMS 345541
Selective allosteric inhibitor of IKK; anti-inflammatory
4809 DSR 6434
Potent TLR7 agonist
4818 PF 04418948
Potent and selective EP2 receptor antagonist
4819 Methylprednisolone
Glucocorticoid receptor agonist
4824 PD 334581
MEK1 inhibitor
4825 TC ASK 10
Potent and selective ASK1 inhibitor; orally bioavailable
4829 ML 239
Breast cancer stem cell inhibitor
4831 NS 3861
α3β2 full agonist; also α3β4 partial agonist
4836 AZ 628
Potent Raf kinase inhibitor
4837 AZD 3988
Potent and selective DGAT-1 inhibitor
4839 AZD 6482
Potent and selective PI 3-Kβ inhibitor
4840 KU 0060648
Dual DNA-PK and PI 3-K inhibitor
4842 BIX 02189
Selective MEK5 and ERK5 inhibitor
4844 HJC 0350
Selective Epac2 inhibitor
4845 A 939572
Potent SCD-1 inhibitor
4847 PluriSln 1
SCD-1 inhibitor
4848 MI 2 (MALT1 inhibitor)
MALT1 inhibitor
4852 Carbetocin
Oxytocin analog
4853 8-pCPT-2-O-Me-cAMP-AM
Selective Epac activator; cell-permeable analog of 8CPT-2Me-cAMP (Cat. No. 1645)
4854 ML 00253764 hydrochloride
Melanocortin MC4 receptor antagonist; brain penetrant
4855 WIKI4
Potent tankyrase inhibitor
4857 Amlexanox
Selective inhibitor of TBK
4860 ML 193
Potent, selective GPR55 antagonist
4862 PPTN hydrochloride
High affinity and selective P2Y14 antagonist
4863 CA 074
Selective cathepsin B inhibitor
4865 APY 29
Inhibits IRE1α autophosphorylation; activates IRE1α endoribonuclease activity
4866 ML 190
Selective κ opioid receptor antagonist
4869 SR 2211
Selective RORγ inverse agonist
4872 KML 29
Highly potent and selective MAGL inhibitor
4874 SR 1078
RORα/γ agonist
4875 Senexin A
Cdk8 inhibitor
4876 Eact
Activator of Ca2+-activated Cl- channel transmembrane protein 16A (TMEM16A)
4877 CaCCinh-A01
Calcium-activated chloride channel (CaCC) inhibitor
4878 H2L5186303
Potent and selective LPA2 receptor antagonist
4879 TC-G 1001
GPR35 agonist; more potent than zaprinast (Cat. No. 0947)
4880 ML 281
STK33 inhibitor
4883 CU CPT 4a
Selective TLR3 inhibitor
4884 CU CPT 22
Selective TLR1/2 inhibitor
4888 KHS 101 hydrochloride
Selective inducer of neuronal differentiation in hippocampal neural progenitors
4889 SGC-CBP30
Potent CBP/p300 BRD inhibitor
4890 AR-C 118925XX
Selective and competitive P2Y2 antagonist
4892 (R)-PFI 2 hydrochloride
Potent and selective SETD7 inhibitor
4894 ML 299
Potent inhibitor of PLD1 and PLD2; CNS penetrant
4897 CYM 5541
Selective S1P3 receptor allosteric agonist
4899 ML 120B dihydrochloride
Novel IKK2-selective inhibitor

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