|
| Cat. No. |
Product Name / Activity |
| 6617 |
LYN 1604 dihydrochloride |
| Potent UNC-51-like kinase 1 (ULK1) agonist |
|
| Cat. No. |
Product Name / Activity |
| 5097 |
A12B4C3 |
| Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor |
| 7283 |
Apilimod dimesylate |
| Potent and selective PIKfyve inhibitor |
| 7511 |
ARN 3236 |
| Potent inhibitor of salt-inducible kinases |
| 7001 |
AT 7867 |
| Potent p70-S6 kinase inhibitor; also potently inhibits Akt and PKA |
| 7673 |
BAY 091 |
| Potent and selective PIP4K2A inhibitor |
| 5123 |
BMX-IN-1 |
| Potent and irreversible BMX inhibitor |
| 5382 |
C16 |
| PKR inhibitor |
| 7018 |
CBR-470-1 |
| PGK1 inhibitor; activates Nrf2 |
| 6558 |
CP 43 |
| Potent TAOK inhibitor |
| 2755 |
DCA |
| Mitochondrial pyruvate dehydrogenase kinase (PDK) inhibitor |
| 7285 |
DCLK1-IN-1 |
| Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable |
| 3572 |
GSK 650394 |
| Serum- and glucocorticoid-regulated kinase (SGK) inhibitor |
| 6976 |
JNJ 10198409 |
| c-Abl, Lck, c-Src and Fyn kinase inhibitor; also inhibits PDGFRα and PDGFRβ |
| 5845 |
JX 06 |
| Potent and selective pyruvate dehydrogenase kinase (PDK) 1/2/3 inhibitor |
| 5604 |
MI 14 |
| Potent and selective PI 4-kinase IIIβ inhibitor |
| 4880 |
ML 281 |
| STK33 inhibitor |
| 5134 |
MRT 67307 dihydrochloride |
| Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor |
| 5780 |
MRT 68921 dihydrochloride |
| ULK inhibitor |
| 7927 |
MSC 1186 |
| Potent and selective SRPK family inhibitor |
| 7371 |
Neratinib |
| Potent inhibitor of MST1; also inhibits EGFR and ErbB2 kinases |
| 5429 |
NG 25 |
| TGF-β-activated kinase (TAK1) inhibitor |
| 3439 |
NH 125 |
| Histidine protein kinase inhibitor; also inhibits CaM kinase III |
| 8175 |
NIBR LTSi New |
| Potent and selective LATS inhibitor; activates YAP signaling |
| 3960 |
NVP 231 |
| Potent, selective and reversible CerK inhibitor |
| 3604 |
(5Z)-7-Oxozeaenol |
| Potent and selective TAK1 MAPKKK inhibitor |
| 5752 |
PF 06260933 dihydrochloride |
| MAP4K4 (HGK) inhibitor; also inhibits MINK and TNIK |
| 4278 |
PF 431396 |
| Dual FAK/PYK2 inhibitor |
| 4630 |
SB 747651A dihydrochloride |
| Potent MSK1 inhibitor; also inhibits other AGC group kinases |
| 6528 |
SGC AAK1 1 |
| AAK1 and BMP2K inhibitor; activates Wnt signaling |
| 6564 |
SGC GAK 1 |
| High affinity cyclin G associated kinase (GAK) inhibitor |
| 5570 |
STOCK2S 26016 |
| Lysine deficient protein kinase (WNK) signaling inhibitor |
| 6430 |
Takinib |
| Potent and selective TAK1/MAP3K7 kinase inhibitor |
| 5240 |
TC-S 7006 |
| Potent and selective Tpl2 (Cot; MAP3K8) inhibitor |
| 3946 |
TNP |
| Inhibitor of IP6K; also inhibits IP3K |
| 5271 |
UNC 3230 |
| Potent and selective PIP5K1C inhibitor; antinociceptive |
| 6604 |
VER 246608 |
| Potent and selective pyruvate dehydrogenase kinase (PDK) 1/2/3/4 inhibitor |
| 5413 |
WH-4-023 |
| Potent salt inducible kinase (SIK) inhibitor; also inhibits Lck and Src |
| 5493 |
XL 413 hydrochloride |
| Potent and selective Cdc7 inhibitor |
| 6482 |
XMU MP 1 |
| Potent and selective MST1/2 inhibitor; orally bioavailable |
|
| Cat. No. |
Product Name / Activity |
| 2600 |
Clofarabine |
| Deoxycytidine kinase (dCK) substrate |
| 6018 |
Nicotinamide Riboside |
| NAD+ precursor; substrate for nicotinamide riboside kinases |
|
| Cat. No. |
Product Name / Activity |
| 7980 |
MTK 458 |
| PINK1 activator |
| 7876 |
PZ 3022 |
| PanK Activator |
| 7809 |
TEPP 46 |
| Potent and selective pyruvate kinase M2 (PKM2) allosteric activator |
|
| Cat. No. |
Product Name / Activity |
| 7425 |
CG 428 |
| Potent tropomyosin receptor kinase (TRK) Degrader |
| 6524 |
TL 12-186 |
| Multikinase Degrader |
|
| Cat. No. |
Product Name / Activity |
| 7426 |
CG 428-Neg |
| Negative control for CG 428 (Cat. No. 7425) |
| 6529 |
SGC AAK1 1N |
| Negative control for SGC AAK1 1 (Cat.No. 6528) |
| 6525 |
TL 13-27 |
| Negative control for TL 12-186 (Cat. No. 6524) |
Other |
| Cat. No. |
Product Name / Activity |
| 7546 |
C28 |
| Potent LMTK3 inhibitor |
| 8122 |
MR 24 New |
| Potent and selective MST3 kinase binding inhibitor |
| 1506 |
Terazosin hydrochloride |
| Increases PGK1 activity; α1 antagonist |